Ianthellamide A, a selective kynurenine-3-hydroxylase inhibitor from the Australian marine sponge Ianthella quadrangulata.

نویسندگان

  • Yunjiang Feng
  • Bruce F Bowden
  • Vimal Kapoor
چکیده

Ianthellamide A (1), a novel octopamine derivative, was isolated from the Australian marine sponge Ianthella quadrangulata. Compound 1 selectively inhibited the activity of kynurenine 3-hydroxylase with an IC(50) value of 1.5 μM. It also significantly increased the level of endogenous kynurenic acid in rat brain and hence has the potential as a neuroprotective agent in the treatment of neurodegenerative disorders.

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عنوان ژورنال:
  • Bioorganic & medicinal chemistry letters

دوره 22 10  شماره 

صفحات  -

تاریخ انتشار 2012